Product Name :
URB-602
Sequence:
Purity:
≥98% (TLC)
Molecular Weight:
295.4
Solubility :
Soluble in DMSO (30 mg/ml) or ethanol (5 mg/ml warm).
Appearance:
Off-white solid.
Use/Stability :
As indicated on product label or CoA when stored as recommended. Store, as supplied, at room temperature for up to 1 year. Store solutions at -20°C for up to 3 months.
Description:
Monoacylglycerol lipase inhibitor Selectively inhibits monoacylglycerol (MAG) lipase (IC50=28µM) via a noncompetitive mechanism.1977557-86-0 Biological Activity Does not inhibit FAAH, DAG lipase or COX-2. URB-602 selectively raises levels of 2-arachidonoylglycerol with no change in anandamide concentrationsin cells and tissues. In the same way anandamide levels were markely elevated by the FAAH inhibitor URB597 at 1µM.
CAS :
565460-15-3
Solubility:
Soluble in DMSO (30 mg/ml) or ethanol (5 mg/ml warm).2492423-29-5 custom synthesis
Formula:
C19H21NO2
Additional Information :
| Alternative Name Biphenyl-3-yl carbamic acid cyclohexyl ester | Appearance Off-white solid.PMID:28722924 | CAS 565460-15-3 | Couple Target Monoacylglycerol lipase | Couple Type Inhibitor | Formula C19H21NO2 | MW 295.4 | MeltingPoint 122-123°C | Purity ≥98% (TLC) | Solubility Soluble in DMSO (30 mg/ml) or ethanol (5 mg/ml warm). | Unit of Measure (UM) mg